Publikationen Dr. Dirk Bier
Journal Article
Preparation and Preclinical Evaluation of 18F-Labeled Olutasidenib Derivatives for Non-Invasive Detection of Mutated Isocitrate Dehydrogenase 1 (mIDH1)
Molecules 29(16), 3939 (2024) [10.3390/molecules29163939]
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Conference Presentation (After Call)
Development and preclinical evaluation of radiofluorinated olutasidenib derivatives for non-invasive detection of mutated isocitrate dehydrogenase 1 (mIDH1) in gliomas
62. Jahrestagung der Deutschen Gesellschaft für Nuklearmedizin, DGN 2024, LeipzigLeipzig, Germany, 10 Apr 2024 - 13 Apr 2024
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Journal Article
Radiosynthesis and In Vitro Evaluation of [11C]tozadenant as Adenosine A2A Receptor Radioligand
Molecules 29(5), 1089 (2024) [10.3390/molecules29051089]
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Journal Article
8-Bicycloalkyl-CPFPX derivatives as potent and selective tools for in vivo imaging of the A1 adenosine receptor
European journal of medicinal chemistry 271, 116380 (2024) [10.1016/j.ejmech.2024.116380]
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Conference Presentation (After Call)
18F-Labelled inhibitors for targeting of IDH1 mutant gliomas
25th International Symposium on Radiopharmaceutical Sciences, ISRS2023, Honolulu, USAHonolulu, USA, USA, 22 May 2023 - 26 May 2023
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Journal Article
AI-based identification of therapeutic agents targeting GPCRs: introducing ligand type classifiers and systems biology
Chemical science 14(32), 8651-8661 (2023) [10.1039/D3SC02352D]
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Conference Presentation (After Call)
F-18-ALX5406: Eine hirngängige Prodrug zur PET-Bildgebung des Glycintransporters Typ 1
60. Jahrestagung der Deutschen Gesellschaft für Nuklearmedizin, LeipzigLeipzig, Germany, 27 Apr 2022 - 30 Apr 2022
[10.1055/s-0042-1745960]
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Conference Presentation (After Call)
Evaluation of a multifunctional blood-brain barrier co-culture model prepared from rat primary brain endothelial cells and astrocytes: first results
24th International Symposium on Radiopharmaceutical Sciences, ISRS2022, NantesNantes, France, 29 May 2022 - 3 Jun 2022
(2022) [10.1016/S0969-8051(22)00233-5]
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Conference Presentation (After Call)
8-Bicycloalkyl-CPFPX derivatives as potent and selective tools for PET imaging of the A1 adenosine receptor
24th International Symposium on Radiopharmaceutical Sciences, ISRS2022, NantesNantes, France, 29 May 2022 - 3 Jun 2022
(2022) [10.1016/S0969-8051(22)00096-8]
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Conference Presentation (After Call)
[18F]ALX5406: a brain-penetrating prodrug for GlyT1-specific PET imaging
24th International Symposium on Radiopharmaceutical Sciences, iSRS 2022, NantesNantes, Germany, 29 May 2022 - 3 Jun 2022
(2022) [10.1016/S0969-8051(22)00127-5]
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Conference Presentation (After Call)
18F-labelled probes for non-invasive assessment of the IDH genotype in diffuse glioma
24th International Symposium on Radiopharmaceutical Sciences, iSRS 2022, NantesNantes, France, 29 May 2022 - 3 Jun 2022
(2022) [10.1016/S0969-8051(22)00081-6]
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Journal Article
[18F]ALX5406: A Brain-Penetrating Prodrug for GlyT1-Specific PET Imaging
ACS chemical neuroscience 12(18), 3335 - 3346 (2021) [10.1021/acschemneuro.1c00284]
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Journal Article
Design, synthesis and biological evaluation of Tozadenant analogues as adenosine A2A receptor ligands
European journal of medicinal chemistry 214, 113214 (2021) [10.1016/j.ejmech.2021.113214]
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Journal Article
Species Differences in Microsomal Metabolism of Xanthine-Derived A1 Adenosine Receptor Ligands
Pharmaceuticals 14(3), 277 - (2021) [10.3390/ph14030277]
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Journal Article
Delivery of the Radionuclide 131I Using Cationic Fusogenic Liposomes as Nanocarriers
International journal of molecular sciences 22(1), 457 - (2021) [10.3390/ijms22010457]
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Journal Article
Preparation of 5-[131I]iodotubercidin for the detection of adenosine kinase
Journal of radioanalytical and nuclear chemistry 326(3), 1691 - 1697 (2020) [10.1007/s10967-020-07465-2]
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Journal Article
Development and Evaluation of a Versatile Receptor-Ligand Binding Assay Using Cell Membrane Preparations Embedded in an Agarose Gel Matrix and Evaluation with the Human Adenosine A1 Receptor
Assay and drug development technologies 18(7), (2020) [10.1089/adt.2020.991]
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Journal Article
Influence of binding affinity and blood plasma level on cerebral pharmacokinetics and PET imaging characteristics of two novel xanthine PET radioligands for the A1 adenosine receptor
Nuclear medicine and biology 82-83, 1 - 8 (2020) [10.1016/j.nucmedbio.2019.12.001]
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Conference Presentation (After Call)
Preparation of [18F]fluoroalkenyliodonium salts and their application for radiolabeling by cross‐coupling reactions
The 23rd International Symposium on Radiopharmaceutical Sciences, BeijingBeijing, China, 26 May 2019 - 31 May 2019
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Journal Article
Relevance of In Vitro Metabolism Models to PET Radiotracer Development: Prediction of In Vivo Clearance in Rats from Microsomal Stability Data
Pharmaceuticals 12(2), 57 (2019) [10.3390/ph12020057]
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Journal Article
Influence of incubation conditions on microsomal metabolism of xanthine-derived A1 adenosine receptor ligands
Journal of pharmacological & toxicological methods 95, 16 - 26 (2019) [10.1016/j.vascn.2018.11.005]
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Journal Article
Synthesis and Pharmacological Evaluation of Identified and Putative Metabolites of the A 1 Adenosine Receptor Antagonist 8-Cyclopentyl-3-(3-fluoropropyl)-1-propylxanthine (CPFPX)
ChemMedChem 12(10), 770 - 784 (2017) [10.1002/cmdc.201600592]
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Journal Article
New potent A1 adenosine receptor radioligands for positron emission tomography
Nuclear medicine and biology 44, 69 - 77 (2017) [10.1016/j.nucmedbio.2016.09.004]
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Journal Article
Efficient synthesis of [$^{18}$ F]FPyME: A new approach for the preparation of maleimide-containing prosthetic groups for the conjugation with thiols
Journal of labelled compounds and radiopharmaceuticals 60(1), 87-92 (2017) [10.1002/jlcr.3469]
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Poster (Plenary/Keynote)
New strategy of a two-step radiosynthesis of [F-18]fluoropyridine-based maleimide-containing prosthetic groups for labelling of peptides and proteins
21st International Symposium on Radiopharmaceutical Sciences, ISRS 2015, ColumbiaColumbia, USA, 26 May 2015 - 31 May 2015
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Conference Presentation (Plenary/Keynote)
Synthesis and in vitro evaluation of radiobrominated adenosine A(1) receptor ligand [*Br] CPBPX
21st International Symposium on Radiopharmaceutical Sciences, ISRS 2015, ColumbiaColumbia, USA, 26 May 2015 - 31 May 2015
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Conference Presentation (Plenary/Keynote)
New metabolically enhanced PET radioligands for the adenosine A(1) receptor
21st International Symposium on Radiopharmaceutical Sciences, ISRS 2015, ColumbiaColumbia, USA, 26 May 2015 - 31 May 2015
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Contribution to a book
Imaging of Adenosine Receptors
PET and SPECT of Neurobiological Systems
Berlin, Heidelberg : Springer Berlin Heidelberg : Chapter 7, 181-198 (2014) [10.1007/978-3-642-42014-6_7]
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Poster (Other)
Synthesis and evaluation of second generation A1 adenosine receptor (A1AR) ligands for PET
20th International Symposium on Radiopharmaceutical Sciences, Jeju IslandJeju Island, Korea, 12 May 2013 - 17 May 2013
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Journal Article
Collision-induced dissociation studies of caffeine in positive electrospray ionisation mass spectrometry using six deuterated isotopomers and one N1-ethylated homologue
Rapid communications in mass spectrometry 27(8), 885 - 895 (2013) [10.1002/rcm.6520]
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Conference Presentation (Other)
Reaction cross section measurements of nachSe(d,xn)75,76,77,78,82Br processes in the energy range 41 -> 17 MeV
7th International Symposium on Radiohalogens, WhistlerWhistler, Canada, 15 Sep 2012 - 19 Sep 2012
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